NVP-BKM120 Hydrochloride - CAS# 1312445-63-8 locaine Hydrochloride Chemical Name: 5-{[7-(benzyloxy)quinazolin-4-yl]amino}-4-fluoro-2-methylphenol
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NVP-BKM120 Hydrochloride - CAS# 1312445-63-8 locaine Hydrochloride Chemical Name: 5-{[7-(benzyloxy)quinazolin-4-yl]amino}-4-fluoro-2-methylphenolBuparlisib, also known as BKM120, is an orally bioavailable specific oral inhibitor of the pan class I phosphatidylinositol 3 kinase (PI3K) family of lipid kinases with potential antineoplastic activity. PI3K inhibitor BKM120 specifically inhibits class I PIK3 in the PI3K AKT kinase (or protein kinase B) signaling pathway in an ATP competitive manner, thereby inhibiting the production of the secondary messenger phosphatidylinositol 3,4,5 trisphosphate
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